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Human prolyl endopeptidase (PREP) - complex with S17092

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Protein Data Bank Japan2026-02-04 更新2026-08-24 收录
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Human prolyl endopeptidase (PREP) - complex with S17092 Descriptor: 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DI(HYDROXYETHYL)ETHER, GLYCEROL, ... Authors: Fucci, I.J, Yoo, E, Monteiro, D.C.F. Deposit date: 2025-08-26 Release date: 2026-01-21 Last modified: 2026-02-04 Method: X-RAY DIFFRACTION (1.81 Å) Cite: Structure-Guided Optimization of 4-Chloro-Pyrazolopyridine Analogs for Covalent PREP Inhibition. J.Med.Chem., 69, 2026

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2025-08-26
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