FGFR-1 in complex with ligand lenvatinib
收藏Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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FGFR-1 in complex with ligand lenvatinib Descriptor: 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide, Fibroblast growth factor receptor 1 Authors: Matsuki, M, Hoshi, T, Yamamoto, Y, Ikemori-Kawada, M, Minoshima, Y, Funahashi, Y, Matsui, J. Deposit date: 2018-05-09 Release date: 2018-07-11 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.86 Å) Cite: Lenvatinib inhibits angiogenesis and tumor fibroblast growth factor signaling pathways in human hepatocellular carcinoma models. Cancer Med, 7, 2018
与配体仑伐替尼(lenvatinib)结合的成纤维细胞生长因子受体1(FGFR-1)。描述物:4-{3-氯-4-[(环丙基氨基甲酰基)氨基]苯氧基}-7-甲氧基喹啉-6-甲酰胺。作者:Matsuki, M、Hoshi, T、Yamamoto, Y、Ikemori-Kawada, M、Minoshima, Y、Funahashi, Y、Matsui, J。存库日期:2018-05-09;发布日期:2018-07-11;最后修改日期:2024-10-16。实验方法:X射线衍射(X-RAY DIFFRACTION,分辨率2.86埃(Å))。引用文献:仑伐替尼可在人类肝细胞癌模型中抑制血管生成与肿瘤成纤维细胞生长因子信号通路,刊载于《癌症医学》(Cancer Med)2018年第7卷。
创建时间:
2018-05-09



