Cyclophosphamide is 4-hydroxylated by CYP2B6
收藏reactome.org2025-01-22 收录
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Cyclophosphamide (CPA) is an alkylating agent used in cancer chemotherapy and an immunosuppressant. CYP2B6 converts CPA to the active metabolite 4-hydroxy-CPA.
环磷酰胺(Cyclophosphamide,简称CPA)作为一种烷化剂,广泛应用于癌症化疗及免疫抑制治疗中。CYP2B6酶能够将环磷酰胺转化为活性代谢产物4-羟基环磷酰胺。
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