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Mycobacterial CIII2CIV2 supercomplex, Inhibitor free

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Protein Data Bank Japan2025-05-14 更新2026-05-23 收录
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Mycobacterial CIII2CIV2 supercomplex, Inhibitor free Descriptor: (2R)-2-(hexadecanoyloxy)-3-{[(S)-hydroxy{[(1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9S)-9-methyloctadecanoate, (2R)-3-(((2-aminoethoxy)(hydroxy)phosphoryl)oxy)-2-(palmitoyloxy)propyl (E)-octadec-9-enoate, (2S)-1-(hexadecanoyloxy)propan-2-yl (10S)-10-methyloctadecanoate, ... Authors: Di Trani, J.M, Yanofsky, D.J, Rubinstein, J.L. Deposit date: 2021-07-16 Release date: 2021-08-04 Last modified: 2025-05-14 Method: ELECTRON MICROSCOPY (3 Å) Cite: Structure of mycobacterial CIII 2 CIV 2 respiratory supercomplex bound to the tuberculosis drug candidate telacebec (Q203). Elife, 10, 2021

分枝杆菌CIII₂CIV₂超级复合物,无抑制剂状态。描述物:(2R)-2-(十六烷酰氧基)-3-{[(S)-羟基{[(1R,2R,3R,4R,5R,6S)-2,3,4,5,6-五羟基环己基]氧基}磷酰基]氧基}丙基 (9S)-9-甲基十八烷酸酯、(2R)-3-(((2-氨基乙氧基)(羟基)磷酰基)氧基)-2-(棕榈酰氧基)丙基 (E)-十八碳-9-烯酸酯、(2S)-1-(十六烷酰氧基)丙-2-基 (10S)-10-甲基十八烷酸酯,……。作者:Di Trani, J.M.、Yanofsky, D.J.、Rubinstein, J.L.。存档日期:2021-07-16;发布日期:2021-08-04;最后修改日期:2025-05-14。研究方法:电子显微镜(分辨率3埃)。引用文献:《结合结核候选药物telacebec(Q203)的分枝杆菌CIII₂CIV₂呼吸超级复合物的结构》,《eLife》,第10卷,2021年。

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2021-07-16
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