PanDDA analysis group deposition -- Aar2/RNaseH in complex with fragment P02C06 from the F2X-Universal Library
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PanDDA analysis group deposition -- Aar2/RNaseH in complex with fragment P02C06 from the F2X-Universal Library Descriptor: 5-methylpyridazin-3(2H)-one, A1 cistron-splicing factor AAR2, Pre-mRNA-splicing factor 8 Authors: Barthel, T, Wollenhaupt, J, Lima, G.M.A, Wahl, M.C, Weiss, M.S. Deposit date: 2022-08-26 Release date: 2022-11-02 Last modified: 2024-05-22 Method: X-RAY DIFFRACTION (1.53 Å) Cite: Large-Scale Crystallographic Fragment Screening Expedites Compound Optimization and Identifies Putative Protein-Protein Interaction Sites. J.Med.Chem., 65, 2022
PanDDA分析团队存档——Aar2/RNaseH与F2X通用文库(F2X-Universal Library)来源的片段P02C06形成的复合物,描述项:5-甲基哒嗪-3(2H)-酮、A1顺式剪接因子(cistron-splicing factor)AAR2、前mRNA剪接因子8(Pre-mRNA-splicing factor 8)。作者:Barthel, T、Wollenhaupt, J、Lima, G.M.A、Wahl, M.C、Weiss, M.S. 存档日期:2022-08-26,发布日期:2022-11-02,最后修改日期:2024-05-22。实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.53埃。引用文献:《大规模晶体学片段筛选加速化合物优化并鉴定潜在蛋白质-蛋白质相互作用位点》,《药物化学杂志(J.Med.Chem.)》,第65卷,2022年
创建时间:
2022-08-26



