Crystal structure of CDK4 in complex with CyclinD1 and P27
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Crystal structure of CDK4 in complex with CyclinD1 and P27 Descriptor: Cyclin-dependent kinase 4, Cyclin-dependent kinase inhibitor 1B, G1/S-specific cyclin-D1 Authors: Guiley, K.Z, Stevenson, J.W, Lou, K, Barkovich, K.J, Bunch, K, Tripathi, S.M, Shokat, K.M, Rubin, S.M. Deposit date: 2019-06-07 Release date: 2019-12-25 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.89 Å) Cite: p27 allosterically activates cyclin-dependent kinase 4 and antagonizes palbociclib inhibition. Science, 366, 2019
CDK4与CyclinD1及P27复合物的晶体结构
描述:细胞周期蛋白依赖性激酶4(Cyclin-dependent kinase 4, CDK4)、细胞周期蛋白依赖性激酶抑制剂1B(Cyclin-dependent kinase inhibitor 1B, p27)、G1/S特异性细胞周期蛋白D1(G1/S-specific cyclin-D1, CyclinD1)
作者:Guiley, K.Z、Stevenson, J.W、Lou, K、Barkovich, K.J、Bunch, K、Tripathi, S.M、Shokat, K.M、Rubin, S.M.
提交日期:2019-06-07
发布日期:2019-12-25
最后更新日期:2024-10-30
实验方法:X射线衍射(分辨率2.89 Å)
引用文献:《p27别构激活细胞周期蛋白依赖性激酶4并拮抗帕博西尼抑制作用》,《科学》,366卷,2019年
创建时间:
2019-06-07



