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Crystal Structure of Danio rerio Histone Deacetylase 10 in Complex with N-methylpiperazine Benzhydroxamic Acid

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Protein Data Bank Japan2024-10-23 更新2026-04-19 收录
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Crystal Structure of Danio rerio Histone Deacetylase 10 in Complex with N-methylpiperazine Benzhydroxamic Acid Descriptor: N-hydroxy-4-[(4-methylpiperazin-1-yl)methyl]benzamide, PHOSPHATE ION, POTASSIUM ION, ... Authors: Herbst-Gervasoni, C.J, Christianson, D.W. Deposit date: 2022-02-27 Release date: 2022-04-06 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Identification of histone deacetylase 10 (HDAC10) inhibitors that modulate autophagy in transformed cells. Eur.J.Med.Chem., 234, 2022

斑马鱼(Danio rerio)组蛋白去乙酰化酶10与N-甲基哌嗪苯并异羟肟酸复合物的晶体结构 描述符:N-羟基-4-[(4-甲基哌嗪-1-基)甲基]苯甲酰胺、磷酸根离子、钾离子…… 作者:Herbst-Gervasoni, C.J.、Christianson, D.W. 沉积日期:2022-02-27 发布日期:2022-04-06 最后修改日期:2024-10-23 检测方法:X射线衍射(分辨率2.1 Å) 引用文献:《调控转化细胞自噬的组蛋白去乙酰化酶10(HDAC10)抑制剂的鉴定》,《欧洲药物化学杂志》,234卷,2022年
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2022-02-27
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