PanDDA analysis group deposition SARS-CoV-2 main protease fragment screen -- Crystal Structure of SARS-CoV-2 main protease in complex with Z1310876699 (Mpro-x0426)
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PanDDA analysis group deposition SARS-CoV-2 main protease fragment screen -- Crystal Structure of SARS-CoV-2 main protease in complex with Z1310876699 (Mpro-x0426) Descriptor: 2-fluoro-N-[2-(pyridin-4-yl)ethyl]benzamide, 3C-like proteinase, DIMETHYL SULFOXIDE Authors: Fearon, D, Owen, C.D, Douangamath, A, Lukacik, P, Powell, A.J, Strain-Damerell, C.M, Resnick, E, Krojer, T, Gehrtz, P, Wild, C, Aimon, A, Brandao-Neto, J, Carbery, A, Dunnett, L, Skyner, R, Snee, M, London, N, Walsh, M.A, von Delft, F. Deposit date: 2020-04-07 Release date: 2020-04-15 Last modified: 2026-02-18 Method: X-RAY DIFFRACTION (1.43 Å) Cite: Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease. Nat Commun, 11, 2020
PanDDA分析小组提交的严重急性呼吸综合征冠状病毒2(SARS-CoV-2)主蛋白酶片段筛选数据集——与配体Z1310876699(Mpro-x0426)结合的SARS-CoV-2主蛋白酶晶体结构。
描述符:2-氟-N-[2-(吡啶-4-基)乙基]苯甲酰胺、3C样蛋白酶(3C-like proteinase)、二甲基亚砜(DIMETHYL SULFOXIDE)
作者:Fearon, D、Owen, C.D、Douangamath, A、Lukacik, P、Powell, A.J、Strain-Damerell, C.M、Resnick, E、Krojer, T、Gehrtz, P、Wild, C、Aimon, A、Brandao-Neto, J、Carbery, A、Dunnett, L、Skyner, R、Snee, M、London, N、Walsh, M.A、von Delft, F.
提交日期:2020-04-07
发布日期:2020-04-15
末次修改日期:2026-02-18
实验方法:X射线衍射(X-RAY DIFFRACTION,分辨率1.43埃)
引用文献:《严重急性呼吸综合征冠状病毒2主蛋白酶的晶体学与亲电片段筛选》,《自然·通讯》,第11卷,2020年
创建时间:
2020-04-07



