Structure of liver pyruvate kinase in complex with anthraquinone derivative 57
收藏Protein Data Bank Japan2024-05-22 更新2026-03-21 收录
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Structure of liver pyruvate kinase in complex with anthraquinone derivative 57 Descriptor: 1,6-di-O-phosphono-beta-D-fructofuranose, 4-amino-3-hydroxy-9,10-dioxo-9,10-dihydroanthracene-2-sulfonic acid, MAGNESIUM ION, ... Authors: Lulla, A, Foller, A, Nain-Perez, A, Grotli, M, Brear, P, Hyvonen, M. Deposit date: 2021-12-01 Release date: 2022-03-16 Last modified: 2024-05-22 Method: X-RAY DIFFRACTION (1.885 Å) Cite: Anthraquinone derivatives as ADP-competitive inhibitors of liver pyruvate kinase. Eur.J.Med.Chem., 234, 2022
与蒽醌衍生物57(anthraquinone derivative 57)结合的肝脏丙酮酸激酶(liver pyruvate kinase)结构 组分:1,6-二-O-磷酰基-β-D-呋喃果糖、4-氨基-3-羟基-9,10-二氧代-9,10-二氢蒽-2-磺酸、镁离子,等
作者:Lulla, A、Foller, A、Nain-Perez, A、Grotli, M、Brear, P、Hyvonen, M
提交日期:2021-12-01
发布日期:2022-03-16
最后修改日期:2024-05-22
实验方法:X射线衍射(分辨率1.885埃)
引用文献:蒽醌衍生物作为肝脏丙酮酸激酶的ADP竞争性抑制剂. 《欧洲药物化学杂志》(Eur.J.Med.Chem.), 234, 2022
创建时间:
2021-12-01



