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Human liver fructose-1,6-bisphosphatase 1 (fructose 1,6-bisphosphate 1-phosphatase, E.C.3.1.3.11) complexed with the allosteric inhibitor 1-(4-bromo-3-methyl-1,2-thiazol-5-yl)-3-(3-methylphenyl)sulfonylurea

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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Human liver fructose-1,6-bisphosphatase 1 (fructose 1,6-bisphosphate 1-phosphatase, E.C.3.1.3.11) complexed with the allosteric inhibitor 1-(4-bromo-3-methyl-1,2-thiazol-5-yl)-3-(3-methylphenyl)sulfonylurea Descriptor: Fructose-1,6-bisphosphatase 1, N-[(4-bromo-3-methyl-1,2-thiazol-5-yl)carbamoyl]-3-methylbenzene-1-sulfonamide Authors: Ruf, A, Joseph, C, Alker, A, Banner, D, Tetaz, T, Benz, J, Kuhn, B, Rudolph, M.G, Yang, H, Shao, C, Burley, S.K. Deposit date: 2017-04-18 Release date: 2019-01-09 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Human liver fructose-1,6-bisphosphatase 1 (fructose 1,6-bisphosphate 1-phosphatase, E.C.3.1.3.11) complexed with the allosteric inhibitor 1-(4-bromo-3-methyl-1,2-thiazol-5-yl)-3-(3-methylphenyl)sulfonylurea To be published

人类肝脏果糖-1,6-二磷酸酶1(fructose 1,6-bisphosphate 1-phosphatase,E.C.3.1.3.11)与变构抑制剂(allosteric inhibitor)1-(4-溴-3-甲基-1,2-噻唑-5-基)-3-(3-甲基苯基)磺酰脲结合形成的复合物。描述符:果糖-1,6-二磷酸酶1,N-[(4-溴-3-甲基-1,2-噻唑-5-基)氨基甲酰]-3-甲基苯-1-磺酰胺。作者:Ruf, A、Joseph, C、Alker, A、Banner, D、Tetaz, T、Benz, J、Kuhn, B、Rudolph, M.G、Yang, H、Shao, C、Burley, S.K。存档日期:2017-04-18;发布日期:2019-01-09;最后修改日期:2024-03-06。实验方法:X射线衍射(X-RAY DIFFRACTION,2.3 Å)。引用文献:人类肝脏果糖-1,6-二磷酸酶1(fructose 1,6-bisphosphate 1-phosphatase,E.C.3.1.3.11)与变构抑制剂1-(4-溴-3-甲基-1,2-噻唑-5-基)-3-(3-甲基苯基)磺酰脲结合形成的复合物,待发表。
创建时间:
2017-04-18
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