Crystal structure of ck1g3 with compound 1
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Crystal structure of ck1g3 with compound 1 Descriptor: 2-[5-methoxy-2-(quinolin-3-yl)pyrimidin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one, Casein kinase I isoform gamma-3, SULFATE ION Authors: Huang, X. Deposit date: 2012-10-08 Release date: 2012-11-21 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Structure-Based Design of Potent and Selective CK1 gamma Inhibitors. ACS Med Chem Lett, 3, 2012
化合物1与CK1γ3的晶体结构
描述项:2-[5-甲氧基-2-(喹啉-3-基)嘧啶-4-基]-1,5,6,7-四氢-4H-吡咯并[3,2-c]吡啶-4-酮、酪蛋白激酶I同工型γ3(Casein kinase I isoform gamma-3)及硫酸根离子
作者:Huang, X.
保藏日期:2012-10-08
发布日期:2012-11-21
最后修改日期:2024-02-28
测试方法:X射线衍射(分辨率2.4 Å)
引用文献:《基于结构设计的强效选择性CK1γ抑制剂》,ACS Med Chem Lett,第3卷,2012年
创建时间:
2012-10-08



