Crystal Structure of SARS-CoV-2 main protease (Nsp5) in complex with compound 17
收藏Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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Crystal Structure of SARS-CoV-2 main protease (Nsp5) in complex with compound 17 Descriptor: 2-cyclobutyl-7-isoquinolin-4-yl-5,7-diazaspiro[3.4]octane-6,8-dione, 3C-like proteinase nsp5 Authors: Talibov, V.O. Deposit date: 2021-04-05 Release date: 2022-02-23 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.23 Å) Cite: Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses. J.Am.Chem.Soc., 144, 2022
新型冠状病毒(SARS-CoV-2)主蛋白酶(Nsp5)与化合物17复合物的晶体结构
配体描述符:2-环丁基-7-异喹啉-4-基-5,7-二氮杂螺[3.4]辛烷-6,8-二酮,3C样蛋白酶nsp5
作者:Talibov, V.O.
提交日期:2021-04-05
发布日期:2022-02-23
最后修改日期:2024-01-31
检测方法:X射线衍射(分辨率2.23 Å)
引用文献:《超大型虚拟筛选发现可广谱抗冠状病毒的新型冠状病毒主蛋白酶抑制剂》,《美国化学会志》,144卷,2022年
创建时间:
2021-04-05



