tRNA guanine Transglycosylase (TGT) in co-crystallized complex with 6-Amino-4-(2-phenylethyl)-1,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one
收藏Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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tRNA guanine Transglycosylase (TGT) in co-crystallized complex with 6-Amino-4-(2-phenylethyl)-1,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one Descriptor: 1,2-ETHANEDIOL, 6-AMINO-4-(2-PHENYLETHYL)-1,7-DIHYDRO-8H-IMIDAZO[4,5-G]QUINAZOLIN-8-ONE, GLYCEROL, ... Authors: Ehrmann, F.R, Nguyen, D, Heine, A, Klebe, G. Deposit date: 2016-02-03 Release date: 2017-02-15 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.89 Å) Cite: Co-crystallization, Isothermal titration calorimetry and nanoESI-MS reveal dimer disturbing inhibitors To be Published
本数据集对应tRNA鸟嘌呤转糖苷酶(tRNA guanine Transglycosylase, TGT)与6-氨基-4-(2-苯乙基)-1,7-二氢-8H-咪唑并[4,5-g]喹唑啉-8-酮的共晶复合物。组分说明:1,2-乙二醇、6-氨基-4-(2-苯乙基)-1,7-二氢-8H-咪唑并[4,5-g]喹唑啉-8-酮、甘油等。作者:Ehrmann F.R.、Nguyen D.、Heine A.、Klebe G.。保藏日期:2016-02-03;发布日期:2017-02-15;最后修改日期:2024-01-10。实验方法:X射线衍射(分辨率1.89埃)。引用文献:《共结晶、等温滴定量热法与纳米电喷雾电离质谱揭示干扰二聚体的抑制剂》(待发表)
创建时间:
2016-02-03



