Crystal Structure of Danio rerio Histone Deacetylase 10 in Complex with Hydroxyethylindole Phenylhydroxamate Inhibitor
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Crystal Structure of Danio rerio Histone Deacetylase 10 in Complex with Hydroxyethylindole Phenylhydroxamate Inhibitor Descriptor: N-hydroxy-4-{[3-(2-hydroxyethyl)-1H-indol-1-yl]methyl}benzamide, PHOSPHATE ION, POTASSIUM ION, ... Authors: Herbst-Gervasoni, C.J, Christianson, D.W. Deposit date: 2020-04-01 Release date: 2020-07-22 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.65 Å) Cite: Structural Basis for the Selective Inhibition of HDAC10, the Cytosolic Polyamine Deacetylase. Acs Chem.Biol., 15, 2020
与羟乙基吲哚苯基异羟肟酸抑制剂结合的斑马鱼(Danio rerio)组蛋白去乙酰化酶10(HDAC10)晶体结构
配体描述:N-羟基-4-{[3-(2-羟乙基)-1H-吲哚-1-基]甲基}苯甲酰胺、磷酸根离子、钾离子及其他组分
作者:Herbst-Gervasoni, C.J.、Christianson, D.W.
保藏日期:2020-04-01
发布日期:2020-07-22
最后修改日期:2024-11-06
实验方法:X射线衍射(2.65埃)
引用文献:《胞质多胺去乙酰化酶HDAC10选择性抑制的结构基础》,发表于Acs Chem.Biol.,第15卷,2020年
创建时间:
2020-04-01



