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Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-Directed Serine Protease Inhibitors

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-Directed Serine Protease Inhibitors Descriptor: 2-(5-{5-[AMINO(IMINIO)METHYL]-1H-BENZIMIDAZOL-2-YL}-2'-FLUORO-6-OXIDO-1,1'-BIPHENYL-3-YL)SUCCINATE, BETA-TRYPSIN, CALCIUM ION, ... Authors: Katz, B.A, Elrod, K, Verner, E, Mackman, R.L, Luong, C, Shrader, W.D, Sendzik, M, Spencer, J.R, Sprengeler, P.A, Kolesnikov, A, Tai, V.W, Hui, H.C, Breitenbucher, J.G, Allen, D, Janc, J.W. Deposit date: 2003-03-06 Release date: 2003-09-02 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.55 Å) Cite: Elaborate manifold of short hydrogen bond arrays mediating binding of active site-directed serine protease inhibitors. J.Mol.Biol., 329, 2003

介导活性位点靶向丝氨酸蛋白酶抑制剂结合的短氢键阵列精密调控体系 描述符:2-(5-{5-[氨基(亚胺鎓)甲基]-1H-苯并咪唑-2-基}-2'-氟-6-氧代-1,1'-联苯-3-基)琥珀酸盐、β-胰蛋白酶(β-trypsin)、钙离子(CALCIUM ION)等 作者:Katz, B.A、Elrod, K、Verner, E、Mackman, R.L、Luong, C、Shrader, W.D、Sendzik, M、Spencer, J.R、Sprengeler, P.A、Kolesnikov, A、Tai, V.W、Hui, H.C、Breitenbucher, J.G、Allen, D、Janc, J.W 入库日期:2003-03-06 发布日期:2003-09-02 最后修改日期:2024-11-13 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.55埃(Å) 引用文献:介导活性位点靶向丝氨酸蛋白酶抑制剂结合的短氢键阵列精密调控体系,《分子生物学杂志》(J.Mol.Biol.),第329卷,2003年
创建时间:
2003-03-06
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