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Crystal structure of human muscle L-lactate dehydrogenase in complex with inhibitor 1, 3-{[3-CARBAMOYL-7-(2,4-DIMETHOXYPYRIMIDIN-5-YL)QUINOLIN-4-YL]AMINO}BENZOIC ACID

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Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Crystal structure of human muscle L-lactate dehydrogenase in complex with inhibitor 1, 3-{[3-CARBAMOYL-7-(2,4-DIMETHOXYPYRIMIDIN-5-YL)QUINOLIN-4-YL]AMINO}BENZOIC ACID Descriptor: 3-{[3-carbamoyl-7-(2,4-dimethoxypyrimidin-5-yl)quinolin-4-yl]amino}benzoic acid, L-lactate dehydrogenase A chain Authors: Kolappan, S, Craig, L. Deposit date: 2014-07-06 Release date: 2014-12-03 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (3.2 Å) Cite: Structures of lactate dehydrogenase A (LDHA) in apo, ternary and inhibitor-bound forms. Acta Crystallogr.,Sect.D, 71, 2015

人类肌肉L-乳酸脱氢酶与抑制剂1(3-{[3-氨基甲酰-7-(2,4-二甲氧基嘧啶-5-基)喹啉-4-基]氨基}苯甲酸)结合的晶体结构。配体描述:3-{[3-氨基甲酰-7-(2,4-二甲氧基嘧啶-5-基)喹啉-4-基]氨基}苯甲酸、L-乳酸脱氢酶A链。作者:Kolappan S、Craig L。沉积日期:2014-07-06。发布日期:2014-12-03。最后修改日期:2024-02-28。实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率3.2埃。引用文献:《无配体(apo)、三元复合物及结合抑制剂形式的乳酸脱氢酶A(LDHA)结构》,发表于《Acta Crystallogr.,Sect.D》2015年第71卷。
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2014-07-06
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