Tetragonal Complex Structure of Protein Kinase CK2 Catalytic Subunit with a Benzotriazole-Based Inhibitor Generated by click-chemistry
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Tetragonal Complex Structure of Protein Kinase CK2 Catalytic Subunit with a Benzotriazole-Based Inhibitor Generated by click-chemistry Descriptor: 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine, CHLORIDE ION, Casein kinase II subunit alpha, ... Authors: Niefind, K, Schnitzler, A, Swider, R, Maslyk, M, Ramos, A. Deposit date: 2015-07-22 Release date: 2015-09-09 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.65 Å) Cite: Synthesis, Biological Activity and Structural Study of New Benzotriazole-Based Protein Kinase CK2 Inhibitors Rsc Adv, 5, 2015
基于点击化学(click-chemistry)描述符构建的蛋白激酶CK2(Protein Kinase CK2)催化亚基与苯并三氮唑类抑制剂的四方复合物结构:4-[4-[2-[4,5,6,7-四溴苯并三氮唑-2-基]乙基]-1,2,3-三氮唑-1-基]丁-1-胺、氯离子、酪蛋白激酶IIα亚基……
作者:Niefind K、Schnitzler A、Swider R、Maslyk M、Ramos A
提交日期:2015-07-22
发布日期:2015-09-09
最后修改日期:2024-01-10
实验方法:X射线衍射(分辨率2.65 Å)
引用文献:《新型苯并三氮唑类蛋白激酶CK2抑制剂的合成、生物活性及结构研究》,Rsc Adv, 5, 2015
创建时间:
2015-07-22



