Crystal structure of human 3-alpha hydroxysteroid dehydrogenase type 3 in complex with NADP+, 5alpha-androstan-3,17-dione and (3beta, 5alpha)-3-hydroxyandrostan-17-one
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Crystal structure of human 3-alpha hydroxysteroid dehydrogenase type 3 in complex with NADP+, 5alpha-androstan-3,17-dione and (3beta, 5alpha)-3-hydroxyandrostan-17-one Descriptor: 4-ANDROSTENE-3-17-DIONE, Aldo-keto reductase family 1 member C2, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... Authors: Zhang, B, Hu, X.-J, Lin, S.-X. Deposit date: 2015-01-16 Release date: 2016-02-17 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Human 3 alpha-hydroxysteroid dehydrogenase type 3: structural clues of 5 alpha-DHT reverse binding and enzyme down-regulation decreasing MCF7 cell growth. Biochem.J., 473, 2016
人类3α-羟类固醇脱氢酶3型与烟酰胺腺嘌呤二核苷酸磷酸(NADP+)、5α-雄烷-3,17-二酮及(3β,5α)-3-羟基雄烷-17-酮结合的晶体结构
描述项:4-雄烯-3,17-二酮、醛酮还原酶家族1成员C2(Aldo-keto reductase family 1 member C2)、烟酰胺腺嘌呤二核苷酸磷酸(NADP),……
作者:Zhang, B、Hu, X.-J、Lin, S.-X.
存档日期:2015年1月16日
发布日期:2016年2月17日
最后修改日期:2024年2月28日
实验方法:X射线衍射(分辨率1.75埃)
引用文献:人类3α-羟类固醇脱氢酶3型:5α-DHT反向结合与酶下调抑制MCF7细胞增殖的结构线索,《生物化学杂志》(Biochem.J.),第473卷,2016年
创建时间:
2015-01-16



