Heteroatom-Guided, Palladium-Catalyzed Regioselective C–H Functionalization in the Synthesis of 3‑Arylquinolines
收藏Figshare2016-02-19 更新2026-04-29 收录
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https://figshare.com/articles/dataset/Heteroatom_Guided_Palladium_Catalyzed_Regioselective_C_H_Functionalization_in_the_Synthesis_of_3_Arylquinolines/2398681
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资源简介:
A new approach for the regioselective functionalization of the C-3-position of quinolines is described. The method utilizes heteroatom guided regioselective C-3 palladation followed by arylation via transmetalation with aryl boronic acids to yield 3-aryl-N-acyl-1,2-dihydroquinolines. In a one-pot sequence, N-deacylation followed by aromatization leads to important 3-arylquinolines in good yields.
创建时间:
2016-02-19



