A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI-CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE
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A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI-CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE Descriptor: 2-(2-HYDROXY-PHENYL)-1H-BENZOIMIDAZOLE-5-CARBOXAMIDINE, ACETYL HIRUDIN, SODIUM ION, ... Authors: Katz, B.A, Elrod, K, Luong, C, Rice, M, Mackman, R.L, Sprengeler, P.A, Spencer, J, Hatayte, J, Janc, J, Link, J, Litvak, J, Rai, R, Rice, K, Sideris, S, Verner, E, Young, W. Deposit date: 2001-01-22 Release date: 2002-01-22 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.75 Å) Cite: A novel serine protease inhibition motif involving a multi-centered short hydrogen bonding network at the active site J.Mol.Biol., 307, 2001
涉及活性位点(active site)处多中心短氢键网络(multi-centered short hydrogen bonding network)的新型丝氨酸蛋白酶(serine protease)抑制基序(inhibition motif)
描述符:2-(2-羟基苯基)-1H-苯并咪唑-5-甲脒、乙酰水蛭素(acetyl hirudin)、钠离子(sodium ion)……
作者:Katz, B.A.、Elrod, K.、Luong, C.、Rice, M.、Mackman, R.L.、Sprengeler, P.A.、Spencer, J.、Hatayte, J.、Janc, J.、Link, J.、Litvak, J.、Rai, R.、Rice, K.、Sideris, S.、Verner, E.、Young, W.
提交日期:2001年1月22日
发布日期:2002年1月22日
最后修改日期:2024年11月13日
实验方法:X射线衍射(X-RAY DIFFRACTION)(1.75 Å)
引用文献:涉及活性位点处多中心短氢键网络的新型丝氨酸蛋白酶抑制基序,J.Mol.Biol.,307卷,2001年
创建时间:
2001-01-22



