CryoEM structure of human 20S proteasome in complex with proteasome inhibitor Salinosporamid A
收藏Protein Data Bank Japan2025-07-02 更新2026-04-19 收录
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CryoEM structure of human 20S proteasome in complex with proteasome inhibitor Salinosporamid A Descriptor: (3AR,6R,6AS)-6-((S)-((S)-CYCLOHEX-2-ENYL)(HYDROXY)METHYL)-6A-METHYL-4-OXO-HEXAHYDRO-2H-FURO[3,2-C]PYRROLE-6-CARBALDEHYDE, Proteasome subunit alpha type-1, Proteasome subunit alpha type-2, ... Authors: Suelzen, H, Boura, E, Silhan, J. Deposit date: 2024-12-09 Release date: 2025-03-05 Last modified: 2025-07-02 Method: ELECTRON MICROSCOPY (2.55 Å) Cite: Structural Insights into Salinosporamide a Mediated Inhibition of the Human 20S Proteasome. Molecules, 30, 2025
人源20S蛋白酶体与蛋白酶体抑制剂Salinosporamid A结合的冷冻电镜(CryoEM)结构
描述符:(3AR,6R,6AS)-6-[(S)-((S)-环己-2-烯基)(羟基)甲基]-6A-甲基-4-氧代-六氢-2H-呋喃并[3,2-c]吡咯-6-甲醛、蛋白酶体亚基α型1、蛋白酶体亚基α型2等
作者:Suelzen H、Boura E、Silhan J
存档日期:2024-12-09
发布日期:2025-03-05
最后修改日期:2025-07-02
实验方法:电子显微镜(分辨率2.55 Å)
引用文献:《Salinosporamide A介导的人源20S蛋白酶体抑制的结构洞察》,发表于《Molecules》,2025年,第30卷
创建时间:
2024-12-09



