Parameters derived from TbrAK kinetics with respect to adenosine in absence and presence of compound 1.

The substrate-inhibition model was applied to fit the raw data; values represent the average of three independently recorded series with each data point measured in triplicate.采用底物抑制模型（substrate-inhibition model）拟合原始实验数据；所有数值为三组独立记录序列的平均值，且每个数据点均进行了三次重复测量。