CRYSTAL STRUCTURE OF AN ACTIVE KRAS G12D (GPPCP) DIMER IN COMPLEX WITH BI-5747
收藏Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF AN ACTIVE KRAS G12D (GPPCP) DIMER IN COMPLEX WITH BI-5747 Descriptor: (3~{S})-5-oxidanyl-3-[2-[[6-[[3-[(1~{S})-6-oxidanyl-3-oxidanylidene-1,2-dihydroisoindol-1-yl]-1~{H}-indol-2-yl]methylamino]hexylamino]methyl]-1~{H}-indol-3-yl]-2,3-dihydroisoindol-1-one, 1,2-ETHANEDIOL, GTPase KRas, ... Authors: Kessler, D. Deposit date: 2020-09-10 Release date: 2020-11-18 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.57 Å) Cite: CRYSTAL STRUCTURE OF AN ACTIVE KRAS G12D (GPPCP) DIMER IN COMPLEX WITH BI-5747 To Be Published
与BI-5747形成复合物的活性KRAS G12D(GPPCP)二聚体的晶体结构
描述项:(3S)-5-羟基-3-[2-[[6-[[3-[(1S)-6-羟基-3-氧代-1,2-二氢异吲哚-1-基]-1H-吲哚-2-基]甲氨基]己基氨基]甲基]-1H-吲哚-3-基]-2,3-二氢异吲哚-1-酮、1,2-乙二醇、GTP酶KRas,……
作者:Kessler, D.
沉积日期:2020-09-10
发布日期:2020-11-18
最后修改日期:2024-01-31
实验方法:X射线衍射(1.57 埃)
引用:与BI-5747形成复合物的活性KRAS G12D(GPPCP)二聚体的晶体结构(待发表)
创建时间:
2020-09-10



