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Crystal Structure of Stabilized Active Plasminogen Activator Inhibitor-1 (PAI-1-stab) in Complex with Two Inhibitory Nanobodies (VHH-2g-42, VHH-2w-64)

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Crystal Structure of Stabilized Active Plasminogen Activator Inhibitor-1 (PAI-1-stab) in Complex with Two Inhibitory Nanobodies (VHH-2g-42, VHH-2w-64) Descriptor: Plasminogen Activator Inhibitor-1, VHH-2g-42, VHH-2w-64 Authors: Sillen, M, Weeks, S.D, Strelkov, S.V, Declerck, P.J. Deposit date: 2018-06-25 Release date: 2020-01-01 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.28 Å) Cite: Molecular mechanism of two nanobodies that inhibit PAI-1 activity reveals a modulation at distinct stages of the PAI-1/plasminogen activator interaction. J.Thromb.Haemost., 18, 2020

稳定型活性纤溶酶原激活物抑制剂-1(Plasminogen Activator Inhibitor-1,PAI-1-stab)与两种抑制性纳米抗体(Nanobodies)(VHH-2g-42、VHH-2w-64)复合物的晶体结构 描述对象:纤溶酶原激活物抑制剂-1、VHH-2g-42、VHH-2w-64 作者:Sillen M、Weeks S.D、Strelkov S.V、Declerck P.J. 提交日期:2018-06-25 发布日期:2020-01-01 最后修改日期:2024-11-13 实验方法:X射线衍射(分辨率2.28埃) 引用文献:两种抑制PAI-1活性的纳米抗体的分子机制揭示了PAI-1与纤溶酶原激活物(Plasminogen Activator)相互作用的不同阶段调控模式。J.Thromb.Haemost., 18, 2020
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2018-06-25
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