Crystal Structure of the first bromodomain of human BRD4 in complex with a triazolo-phthalazine ligand
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Crystal Structure of the first bromodomain of human BRD4 in complex with a triazolo-phthalazine ligand Descriptor: 2-chloro-N-[5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)-2-(morpholin-4-yl)phenyl]benzenesulfonamide, Bromodomain-containing protein 4, SUCCINIC ACID Authors: Filippakopoulos, P, Picaud, S, Felletar, I, Martin, S, Fedorov, O, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2013-11-25 Release date: 2013-12-18 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (1.58 Å) Cite: Crystal Structure of the first bromodomain of human BRD4 in complex with a triazolo-phthalazine ligand To be Published
人BRD4首个溴结构域（bromodomain）与三唑并酞嗪配体复合物的晶体结构
配体描述：2-氯-N-[5-(3-甲基[1,2,4]三唑并[3,4-a]酞嗪-6-基)-2-(吗啉-4-基)苯基]苯磺酰胺；含溴结构域蛋白4（Bromodomain-containing protein 4）；琥珀酸
作者：Filippakopoulos, P、Picaud, S、Felletar, I、Martin, S、Fedorov, O、von Delft, F、Arrowsmith, C.H、Edwards, A.M、Bountra, C、Knapp, S、结构基因组联盟（Structural Genomics Consortium, SGC）
提交日期：2013-11-25
发布日期：2013-12-18
最后修改日期：2024-02-28
研究方法：X射线衍射（X-RAY DIFFRACTION，分辨率1.58埃（Å））
引用文献：人BRD4首个溴结构域与三唑并酞嗪配体复合物的晶体结构 待发表
创建时间：
2013-11-25
