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Structure of human PARP1 catalytic domain bound to a quinazoline-2,4(1H,3H)-dione inhibitor

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Protein Data Bank Japan2024-03-20 更新2026-03-21 收录
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Structure of human PARP1 catalytic domain bound to a quinazoline-2,4(1H,3H)-dione inhibitor Descriptor: 1-[[3-(4-ethyl-3-oxidanylidene-piperazin-1-yl)carbonyl-4-fluoranyl-phenyl]methyl]quinazoline-2,4-dione, Poly [ADP-ribose] polymerase 1 Authors: Cao, R, Wang, Y.L, Zhou, J, Yao, H.P, Huang, N, Xu, B.L. Deposit date: 2016-07-05 Release date: 2016-12-21 Last modified: 2024-03-20 Method: X-RAY DIFFRACTION (2.65 Å) Cite: Structure of human PARP1 catalytic domain bound to a quinazoline-2,4(1H,3H)-dione inhibitor To Be Published

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2016-07-05
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