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Crystal structure of PPAR gamma (PPARG) in complex with SA112 (compound 2).

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Protein Data Bank Japan2024-02-07 更新2026-05-23 收录
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Crystal structure of PPAR gamma (PPARG) in complex with SA112 (compound 2). Descriptor: 2-[4-chloranyl-6-[[3-(2-phenylethoxy)phenyl]amino]pyrimidin-2-yl]sulfanylethanoic acid, GLYCEROL, Peroxisome proliferator-activated receptor gamma Authors: Chaikuad, A, Arifi, S, Merk, D, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2022-08-24 Release date: 2023-07-12 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPAR gamma Modulation. J.Am.Chem.Soc., 145, 2023
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2022-08-24
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