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PAK4 in complex with compound 7

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Protein Data Bank Japan2025-07-16 更新2026-05-23 收录
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https://pdbj.org/mine/summary/9d53
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PAK4 in complex with compound 7 Descriptor: N~2~-{[(1s,4s)-4-aminocyclohexyl]methyl}-N~4~-(5-cyclopropyl-1,3-thiazol-2-yl)pyrimidine-2,4-diamine, Serine/threonine-protein kinase PAK 4 Authors: Boone, C.D, Olland, A.M, Suto, R.K. Deposit date: 2024-08-13 Release date: 2025-04-02 Last modified: 2025-07-16 Method: X-RAY DIFFRACTION (2.468 Å) Cite: Identification of a p21-activated kinase 1 (PAK1) inhibitor with 10-fold selectivity against PAK2. Bioorg.Med.Chem.Lett., 127, 2025
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2024-08-13
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