Corticotropin-releasing hormone receptor 1(CRF1R) bound with BMK-C205 by XFEL

Corticotropin-releasing hormone receptor 1(CRF1R) bound with BMK-C205 by XFEL Descriptor: 8-(4-bromanyl-2,6-dimethoxy-phenyl)-~{N}-butyl-~{N}-(cyclopropylmethyl)-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-4-amine, Endolysin, Isoform CRF-R2 of Corticotropin-releasing factor receptor 1, ... Authors: Cho, H.S, Kim, H. Deposit date: 2022-09-08 Release date: 2023-09-13 Last modified: 2026-03-04 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Structure-based drug discovery of a corticotropin-releasing hormone receptor 1 antagonist using an X-ray free-electron laser. Exp.Mol.Med., 55, 2023