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Crystal structure of DCLK1 kinase domain in complex with ruxolitinib

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Protein Data Bank Japan2023-11-29 更新2026-04-19 收录
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Crystal structure of DCLK1 kinase domain in complex with ruxolitinib Descriptor: (3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile, Isoform 4 of Serine/threonine-protein kinase DCLK1 Authors: Lim, H.J, Jang, D.M, Kim, H.S. Deposit date: 2021-06-16 Release date: 2021-08-18 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Structural Basis of Inhibition of DCLK1 by Ruxolitinib. Int J Mol Sci, 22, 2021

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2021-06-16
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