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Crystal Structure of Aurora2 kinase in complex with a GSK3beta inhibitor

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Protein Data Bank Japan2023-09-06 更新2026-03-21 收录
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Crystal Structure of Aurora2 kinase in complex with a GSK3beta inhibitor Descriptor: N-[6-(4-hydroxyphenyl)-1H-indazol-3-yl]butanamide, Serine/threonine-protein kinase 6 Authors: Maignan, S, Guilloteau, J.P, Pouzieux, S. Deposit date: 2010-01-07 Release date: 2010-03-02 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Rational design of potent GSK3beta inhibitors with selectivity for Cdk1 and Cdk2. Bioorg.Med.Chem.Lett., 20, 2010

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2010-01-07
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