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Kinase domain of MERTK in complex with compound 8

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Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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Kinase domain of MERTK in complex with compound 8 Descriptor: 1,2-ETHANEDIOL, 2-[[2,5-bis(fluoranyl)phenyl]methylamino]-4-(cyclopentylamino)-N-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide, Tyrosine-protein kinase Mer Authors: Schroeder, M, Russ, N, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2021-04-19 Release date: 2021-05-19 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.65 Å) Cite: Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase. J.Med.Chem., 64, 2021

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2021-04-19
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