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Crystal structure of Protein Kinase A in complex with Pyridine-Pyrazolopyridine Based Inhibitors

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Protein Data Bank Japan2023-12-27 更新2026-03-21 收录
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Crystal structure of Protein Kinase A in complex with Pyridine-Pyrazolopyridine Based Inhibitors Descriptor: (2S)-1-{[5-(1H-INDAZOL-5-YL)PYRIDIN-3-YL]OXY}-3-[(7AS)-7AH-INDOL-3-YL]PROPAN-2-AMINE, Inhibitory peptide, cAMP-dependent protein kinase, ... Authors: Stoll, V.S. Deposit date: 2007-01-09 Release date: 2007-03-20 Last modified: 2023-12-27 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Design and synthesis of pyridine-pyrazolopyridine-based inhibitors of protein kinase B/Akt. Bioorg.Med.Chem., 15, 2007

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2007-01-09
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