RORy in complex with inverse agonist 3.
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RORy in complex with inverse agonist 3. Descriptor: 1-methyl-~{N}-(1-thiophen-2-ylcarbonyl-3,4-dihydro-2~{H}-quinolin-6-yl)-~{N}-[2,2,2-tris(fluoranyl)ethyl]indole-4-sulfonamide, Nuclear receptor ROR-gamma Authors: Marcotte, D.M. Deposit date: 2015-11-17 Release date: 2016-04-27 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.803 Å) Cite: Discovery of biaryls as ROR gamma inverse agonists by using structure-based design. Bioorg.Med.Chem.Lett., 26, 2016
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2015-11-17



