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X-ray structure of human PPAR alpha ligand binding domain-seladelpar co-crystals obtained by cross-seeding

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Protein Data Bank Japan2023-09-06 更新2026-05-23 收录
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X-ray structure of human PPAR alpha ligand binding domain-seladelpar co-crystals obtained by cross-seeding Descriptor: GLYCEROL, Peroxisome proliferator-activated receptor alpha, Seladelpar Authors: Kamata, S, Honda, A, Machida, Y, Uchii, K, Shiiyama, Y, Masuda, R, Iino, S, Oyama, T, Ishii, I. Deposit date: 2022-12-24 Release date: 2023-08-09 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (2.01 Å) Cite: Functional and Structural Insights into the Human PPAR alpha / delta / gamma Targeting Preferences of Anti-NASH Investigational Drugs, Lanifibranor, Seladelpar, and Elafibranor. Antioxidants, 12, 2023

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2022-12-24
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