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Notum Inhibitor ARUK3004903

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Protein Data Bank Japan2024-10-16 更新2026-04-19 收录
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Notum Inhibitor ARUK3004903 Descriptor: 1,2-ETHANEDIOL, 1-[3,4-bis(chloranyl)-5-methyl-indol-1-yl]ethanone, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... Authors: Zhao, Y, Jones, E.Y, Fish, P. Deposit date: 2022-11-28 Release date: 2022-12-14 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.4 Å) Cite: Designed switch from covalent to non-covalent inhibitors of carboxylesterase Notum activity. Eur.J.Med.Chem., 251, 2023

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2022-11-28
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