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Protein kinase MKK7 in complex with cyclobutyl-substituted indazole

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Protein Data Bank Japan2024-11-13 更新2026-03-28 收录
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Protein kinase MKK7 in complex with cyclobutyl-substituted indazole Descriptor: Dual specificity mitogen-activated protein kinase kinase 7, ~{N}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{H}-indazol-3-yl)-5-(propanoylamino)benzamide Authors: Buehrmann, M, Wiese, J.N, Mueller, M.P, Rauh, D. Deposit date: 2021-06-15 Release date: 2022-07-20 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Optimization of Covalent MKK7 Inhibitors via Crude Nanomole-Scale Libraries. J.Med.Chem., 65, 2022

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2021-06-15
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