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Crystal structure of MLLT1 (ENL) YEATS domain in complexed with compound 94

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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Crystal structure of MLLT1 (ENL) YEATS domain in complexed with compound 94 Descriptor: 1,2-ETHANEDIOL, 1-cyclopropyl-~{N}-[2-[[(2~{S})-2-methylpyrrolidin-1-yl]methyl]-3~{H}-benzimidazol-5-yl]indazole-5-carboxamide, Protein ENL, ... Authors: Heidenreich, D, Chaikuad, A, Moustakim, M, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Fedorov, O, Brennan, P.E, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2018-10-02 Release date: 2018-10-17 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Discovery of an MLLT1/3 YEATS Domain Chemical Probe. Angew. Chem. Int. Ed. Engl., 57, 2018

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2018-10-02
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