Cryo-EM reconstruction of zampanolide-bound microtubule
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Cryo-EM reconstruction of zampanolide-bound microtubule Descriptor: (2Z,4E)-N-[(S)-[(1S,2E,5S,8E,10Z,17S)-3,11-dimethyl-19-methylidene-7,13-dioxo-6,21-dioxabicyclo[15.3.1]henicosa-2,8,10-trien-5-yl](hydroxy)methyl]hexa-2,4-dienamide, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ... Authors: Kellogg, E.H, Hejab, N.M.A, Nogales, E. Deposit date: 2016-08-11 Release date: 2017-02-01 Last modified: 2024-03-06 Method: ELECTRON MICROSCOPY (3.5 Å) Cite: Insights into the Distinct Mechanisms of Action of Taxane and Non-Taxane Microtubule Stabilizers from Cryo-EM Structures. J. Mol. Biol., 429, 2017
结合扎诺拉利德(zampanolide)的微管的冷冻电镜(Cryo-EM)三维重构结构。 描述项:(2Z,4E)-N-[(S)-[(1S,2E,5S,8E,10Z,17S)-3,11-二甲基-19-亚甲基-7,13-二氧代-6,21-二氧杂双环[15.3.1]二十一碳-2,8,10-三烯-5-基(羟基)甲基]己-2,4-二烯酰胺、鸟苷-5'-二磷酸(GUANOSINE-5'-DIPHOSPHATE)、鸟苷-5'-三磷酸(GUANOSINE-5'-TRIPHOSPHATE)等。 作者:Kellogg, E.H.、Hejab, N.M.A.、Nogales, E. 存档日期:2016-08-11 发布日期:2017-02-01 最后修改日期:2024-03-06 实验方法:电子显微镜(ELECTRON MICROSCOPY),分辨率3.5 Å 引用文献:《基于冷冻电镜结构解析紫杉烷与非紫杉烷类微管稳定剂的独特作用机制》,《Journal of Molecular Biology》,2017年,第429卷。



