遇见数据集

BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-BISAMIDE

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-BISAMIDE Descriptor: 2,2'-oxybis(N-{[4-(3-{2,6-difluoro-3-[(propane-1-sulfonyl)amino]benzoyl}-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl]methyl}acetamide), BENZAMIDINE, Serine/threonine-protein kinase B-raf Authors: Grasso, M.J, Marmorstein, R. Deposit date: 2016-05-09 Release date: 2016-09-14 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.702 Å) Cite: Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAF(V600E) Conformation. Acs Chem.Biol., 11, 2016

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2016-05-09
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