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Irreversible Mcl-1/HIT2 Complex

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Protein Data Bank Japan2025-12-10 更新2026-05-23 收录
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Irreversible Mcl-1/HIT2 Complex Descriptor: (1R)-N-{5-[(dihydroxy-lambda~4~-sulfanyl)oxy]pyridin-3-yl}-2,3-dihydro-1H-indene-1-carboxamide, Induced myeloid leukemia cell differentiation protein Mcl-1 Authors: Muzzarelli, K.M, Assar, Z, Udompholkul, P, Pellecchia, M, Baggio, C, Prentiss, A.M. Deposit date: 2024-11-20 Release date: 2025-11-19 Last modified: 2025-12-10 Method: X-RAY DIFFRACTION (1.82 Å) Cite: A Fragment-Based Electrophile-First Approach to Target Histidine with Aryl-Fluorosulfates: Application to hMcl-1. J.Med.Chem., 68, 2025

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2024-11-20
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